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He aha ʻo Macitentan a me Tadalafil: Nā hoʻohana, ka nui, nā hopena ʻaoʻao a me nā mea hou aku

Created at:1/13/2025

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ʻO Macitentan a me tadalafil he lāʻau lapaʻau hui pū e kōkua ana i ka mālama ʻana i ka maʻi hypertension arterial pulmonary (PAH), kahi maʻi koʻikoʻi kahi e lilo ai ke koko i loko o kou māmā i ke kiʻekiʻe weliweli. Hoʻohui kēia ala lapaʻau ʻelua i ʻelua mau lāʻau lapaʻau like ʻole e hana pū ana e wehe i kou mau kīʻaha koko māmā a hoʻomaikaʻi i ke kahe koko.

Ke loaʻa iā ʻoe ka PAH, e ʻuʻuku a paʻakikī nā ʻaʻa liʻiliʻi i loko o kou māmā, e hana nui ana kou puʻuwai e pauma i ke koko ma o lākou. Hoʻoponopono kēia lāʻau lapaʻau hui i ka pilikia mai nā kihi ʻelua, e hāʻawi ana iā ʻoe i kahi ala lapaʻau piha aʻe ma mua o ka hoʻohana ʻana i kekahi lāʻau.

He aha ʻo Macitentan a me Tadalafil?

Hoʻohui kēia lāʻau lapaʻau i ʻelua mau mea hana e kuhikuhi ana i nā ala like ʻole i loko o kou kino e mālama ai i ka hypertension arterial pulmonary. Kāohi ʻo Macitentan i kekahi mau mea hoʻokipa e hoʻoulu ai i nā kīʻaha koko, ʻoiai ʻo tadalafil e kōkua i ka hoʻomaha ʻana i ka ʻiʻo maʻemaʻe i loko o kou mau paia kīʻaha koko.

Hele mai ka hui ʻana ma ke ʻano o nā papa waha āu e lawe ai ma ka waha, maʻamau i hoʻokahi manawa i ka lā. Kauoha kāu kauka i kēia ke hāʻawi ʻole ka lāʻau lapaʻau hoʻokahi i ka pono lawa, a i ʻole ke koi ʻana o kou maʻi i kahi ala lapaʻau ʻoi aku ka ikaika mai ka hoʻomaka.

Ua aʻo nui ʻia nā mea ʻelua ma kā lākou iho a me ka hui pū ʻana, e hōʻike ana e hiki ke ʻoi aku ka maikaʻi o ka hui ʻana ma mua o kekahi lāʻau i hoʻohana ʻia no ka mālama ʻana i nā hōʻailona PAH a me ka hoʻolohi ʻana i ka holomua o ka maʻi.

No ke aha e hoʻohana ʻia ai ʻo Macitentan a me Tadalafil?

Hoʻolālā ʻia kēia lāʻau lapaʻau hui e mālama i ka hypertension arterial pulmonary, kahi maʻi kakaʻikahi akā koʻikoʻi e pili ana i nā ʻaʻa i loko o kou māmā. Hoʻopilikia ka PAH i ke kahe ʻana o ke koko ma kou māmā, e hoʻokau ana i ke koʻikoʻi ma ka ʻaoʻao ʻākau o kou puʻuwai.

Hiki i kāu kauka ke kuhikuhi i kēia hui inā ʻoe e ʻike nei i nā hōʻailona e like me ka pōkole o ka hanu i ka wā o nā hana o kēlā me kēia lā, ka ʻeha o ka umauma, ka luhi, a i ʻole ka pehu ʻana i kou mau wāwae a me nā kuʻekuʻe wāwae. Hiki mai kēia mau hōʻailona no ka mea e hana nui ana kou puʻuwai e pauma i ke koko ma nā ʻaʻa māmā i hoʻopaʻa ʻia.

Kōkua ka lāʻau lapaʻau i ka hoʻomaikaʻi ʻana i kou hiki ke hoʻoikaika kino, ʻo ia hoʻi hiki iā ʻoe ke hele i kahi mamao a hana i nā hana hou aku me ka ʻole e hanu. Kōkua nō hoʻi ia i ka hoʻolohi ʻana i ka holomua o ka PAH, e hōʻemi ana i kou pilikia o ka hoʻopaʻa ʻia ʻana i ka haukapila a me nā pilikia koʻikoʻi ʻē aʻe.

Pehea e hana ai ʻo Macitentan a me Tadalafil?

Hana kēia hui lāʻau lapaʻau ma o nā ʻano hana ʻelua like ʻole e hāʻawi i ka mālama piha no kou hypertension arterial pulmonary. E noʻonoʻo iā ia e like me ka hoʻoponopono ʻana i ka pilikia mai nā kihi he nui e hāʻawi iā ʻoe i nā hopena maikaʻi aʻe.

Pale ʻo Macitentan i nā mea loaʻa endothelin i loko o kou mau kīʻaha koko. He mea ka endothelin e hoʻopaʻa ai a hoʻopaʻa i nā kīʻaha koko, no laila ma ka pale ʻana i kēia mau mea loaʻa, kōkua ʻo macitentan i ka mālama ʻana i kou mau ʻaʻa māmā e wehe a hoʻomaha.

Hana ʻo Tadalafil ma ka pale ʻana i kahi enzyme i kapa ʻia ʻo PDE5, e alakaʻi ana i ka piʻi ʻana o nā pae o kahi mea e kōkua ai i nā kīʻaha koko e hoʻomaha. Hoʻokumu kēia i kahi kahe koko maʻalahi ma kou mau ʻaʻa māmā a hoʻemi i ke kaomi e kū ana kou puʻuwai.

ʻO ka hui pū ʻana, hana kēia mau lāʻau lapaʻau i kahi hopena synergistic, ʻo ia hoʻi, hana lākou i ka maikaʻi ma mua o ka hana ʻana i ka ʻokoʻa. Manaʻo ʻia kēia ʻano hui he ikaika iki a mālama ʻia no nā maʻi e pono ai ka mālama piha.

Pehea wau e lawe ai iā Macitentan a me Tadalafil?

E lawe i kēia lāʻau lapaʻau e like me ke kauoha a kāu kauka, maʻamau i hoʻokahi manawa i ka lā me ka ʻole o ka meaʻai. Hiki iā ʻoe ke lawe me ka wai, a ʻaʻole ia he mea nui inā ʻoe e ʻai ma mua a ma hope paha o ka lawe ʻana i kāu mahele.

E hoʻāʻo e lawe i kāu lāʻau i ka manawa like i kēlā me kēia lā e mālama i nā pae paʻa i loko o kou kahe koko. Kōkua kēia i ka hōʻoia ʻana i ka mālama mau ʻana i kou maʻi hypertension pulmonary arterial i ka lā.

E ale i ka papa holoʻokoʻa me ka ʻole o ka ʻoki ʻana, ka wāwahi ʻana, a i ʻole ka nau ʻana. Inā pilikia ʻoe i ka ale ʻana i nā pila, e kamaʻilio me kāu kauka e pili ana i nā koho ʻē aʻe a i ʻole nā ʻenehana e kōkua ai.

Mai hooki i ka lawe ʻana i kēia lāʻau lapaʻau i ka wā koke, ʻoiai inā ʻoe e maikaʻi ana. He maʻi maʻi ʻo PAH e pono ai ka mālama mau ʻana, a ʻo ka hooki ʻana i ka wā koke e hiki ke hoʻonui i kou mau hōʻailona.

Pehea ka lōʻihi e lawe ai au i ka Macitentan a me Tadalafil?

He lapaʻau lōʻihi kēia e pono ai ʻoe e hoʻomau i ka wā e kōkua ana i ka mālama ʻana i kou maʻi hypertension pulmonary arterial. He maʻi maʻi ʻo PAH ʻaʻole e hele wale, no laila pono ka lāʻau lapaʻau mau.

E nānā kāu kauka i kāu pane ʻana i ka lāʻau lapaʻau ma o nā nānā maʻamau, me nā hoʻokolohua e ana i kou hiki ke hoʻoikaika kino a me ka hana o ka naʻau. Kōkua kēia mau manawa e hoʻoholo inā e hana maikaʻi ana ka lāʻau lapaʻau iā ʻoe a inā pono e hana i nā hoʻoponopono.

Pono paha kekahi poʻe maʻi e lawe i kēia hui ʻana no nā makahiki, a ʻo nā mea ʻē aʻe e hoʻololi i nā lāʻau lapaʻau like ʻole ma muli o ke ʻano o kā lākou maʻi. E hoʻopilikino ʻia kāu hoʻolālā lapaʻau ma muli o kāu mau pono kikoʻī a me ka maikaʻi o kou ʻae ʻana i ka lāʻau lapaʻau.

He aha nā hopena ʻaoʻao o Macitentan a me Tadalafil?

E like me nā lāʻau lapaʻau a pau, hiki i kēia hui ʻana ke hoʻoulu i nā hopena ʻaoʻao, ʻoiai ʻaʻole ʻike nā mea a pau iā lākou. Hiki ke mālama ʻia ka hapa nui o nā hopena ʻaoʻao a ʻoi aku ka maikaʻi i ka wā e hoʻoponopono ai kou kino i ka lāʻau lapaʻau.

Eia nā hopena ʻaoʻao maʻamau e ʻike ai ʻoe i ka wā e hoʻoponopono ai kou kino i kēia lapaʻau:

  • ʻEha poʻo, e maikaʻi pinepine ana ma hope o nā pule mua
  • ʻUlaʻula a i ʻole ka manaʻo mehana ma kou maka a me kou ʻāʻī
  • Pehu i kou mau wāwae, nā kuʻekuʻe wāwae, a i ʻole nā wāwae
  • Paʻa ihu a i ʻole ka ihu paʻa
  • Hōʻeha ʻōpū a i ʻole ka maʻi
  • Pōniuniu, ʻoiai ke kū koke ʻana
  • ʻEha kua a i ʻole nā ʻeha ʻiʻo

E maʻa mau ana kēia mau hopena ʻaoʻao maʻamau i ka wā, akā e haʻi i kāu kauka inā mau lākou a i ʻole e hoʻopilikia i kāu mau hana i kēlā me kēia lā.

Pono kekahi mau hopena ʻaoʻao koʻikoʻi i ka lāʻau lapaʻau koke, ʻoiai ʻaʻole maʻamau lākou. E kelepona koke i kāu kauka inā ʻike ʻoe i kekahi o kēia mau hōʻailona e pili ana:

  • Nā loli ʻike koke a i ʻole ka nalowale o ka ʻike
  • Nalowale lohe koke a i ʻole ke kani ʻana i kou mau pepeiao
  • ʻEha umauma a i ʻole ka puʻuwai ʻole
  • Pōniuniu nui a i ʻole ka hāʻule
  • Nā hōʻailona o nā pilikia o ke akepaʻa e like me ka melemele o ka ʻili a i ʻole nā maka
  • ʻO ka hanu ʻole maʻamau a i ʻole ka hanu ʻino
  • ʻO ka kū ʻana o ka ʻeha e mau ana ma mua o 4 mau hola (no nā kāne)

He kakaikahi kēia mau hopena ʻaoʻao koʻikoʻi, akā he mea nui e ʻike iā lākou i ka wā mua i hiki ai iā ʻoe ke loaʻa ka mālama olakino kūpono inā pono.

ʻO wai ka mea ʻaʻole pono e lawe iā Macitentan a me Tadalafil?

ʻAʻole kūpono kēia lāʻau lapaʻau hui ʻana no nā mea a pau, a e nānā pono kāu kauka i kāu moʻolelo olakino ma mua o ke kau ʻana. Hiki i kekahi mau maʻi a me nā lāʻau lapaʻau ke palekana ʻole a i ʻole ka liʻiliʻi o kēia lapaʻau.

ʻAʻole pono ʻoe e lawe i kēia lāʻau lapaʻau inā e hoʻohana nei ʻoe i nā lāʻau nitrate no ka ʻeha umauma, no ka mea, hiki i kēia hui ʻana ke hoʻohaʻahaʻa i ke koko. Aia i loko o kēia nā nitrates kauoha e like me ka nitroglycerin a me nā lāʻau leʻaleʻa i kapa ʻia ʻo "poppers."

Pono nā wahine e hāpai ana a i ʻole e hoʻāʻo nei e hāpai e pale i kēia lāʻau lapaʻau, no ka mea, hiki iā ia ke hana i nā kīnā hānau koʻikoʻi. Inā hāpai ʻoe i ka wā e lawe ana i kēia lāʻau lapaʻau, e kelepona koke i kāu kauka e kūkākūkā i nā koho palekana.

ʻAʻole paha e kūpono nā kānaka me ka maʻi ate koʻikoʻi a i ʻole nā maʻi puʻuwai kekahi i kēia lapaʻau. E loiloi kāu kauka i kāu hana ate a me ke olakino o ka puʻuwai ma mua o ka hoʻomaka ʻana iā ʻoe i kēia lāʻau.

Inā he moʻolelo kou o nā pilikia ʻike, ka nalowale o ka lohe, a i ʻole ke koko haʻahaʻa, pono kāu kauka e loiloi pono i nā pōmaikaʻi a me nā pilikia ma mua o ke kau ʻana i kēia hui pū ʻana.

Nā inoa inoa Macitentan a me Tadalafil

Loaʻa kēia lāʻau hui pū ʻia ma lalo o ka inoa inoa ʻo Opsynvi, ʻo ia ka mea i hana nui ʻia i ʻae ʻia no ka mālama ʻana i ka pulmonary arterial hypertension. Kōkua ka inoa inoa i ka hoʻokaʻawale ʻana mai nā lāʻau ʻē aʻe i loaʻa kēia mau mea i nā ʻāpana.

Hiki nō hoʻi iā ʻoe ke hālāwai me nā mea i kūʻai ʻia i nā inoa inoa like ʻole. Loaʻa ʻo Macitentan ma ke ʻano he Opsumit, a ʻike ʻia ʻo tadalafil e nā inoa inoa like ʻole me Cialis a me Adcirca.

E hoʻohana mau i ka inoa inoa a me ka hana i kauoha ʻia e kāu kauka, no ka mea, hiki i nā hana like ʻole ke loaʻa nā ikaika like ʻole a i ʻole nā ʻano hoʻokuʻu e pili ana i ka maikaʻi o ka hana ʻana o ka lāʻau no kou maʻi.

Nā koho ʻē aʻe o Macitentan a me Tadalafil

Nui nā lapaʻau ʻē aʻe no ka pulmonary arterial hypertension inā ʻaʻole kūpono kēia hui pū ʻana iā ʻoe a i ʻole ʻaʻole e hāʻawi i ka mana o nā hōʻailona. Hiki i kāu kauka ke kōkua i ka hoʻoholo ʻana i ke koho e hana maikaʻi loa no kāu kūlana.

ʻO nā lāʻau lapaʻau waha ʻē aʻe no PAH me bosentan, ambrisentan, sildenafil, a me riociguat. Hana kēlā me kēia mea ma nā ala like ʻole e kōkua ai i ka wehe ʻana i nā kīʻaha koko o kou māmā a hoʻemi i ke kaomi pulmonary.

No nā hihia koʻikoʻi, hiki i kāu kauka ke noʻonoʻo i nā lāʻau lapaʻau i hoʻokomo ʻia a i ʻole intravenous e like me epoprostenol, treprostinil, a i ʻole iloprost. Hoʻokaʻawale ʻia kēia mau lapaʻau no nā maʻi me ka maʻi holomua a i ʻole ka poʻe i pane ʻole i nā lāʻau lapaʻau waha.

Loaʻa i kekahi poʻe maʻi ka pōmaikaʻi mai ka hui pū ʻana o nā lāʻau lapaʻau like ʻole, aʻo nā mea ʻē aʻe e maikaʻi me ka lāʻau lapaʻau ma ke kaʻina, kahi e hoʻohui ʻia ai nā lāʻau lapaʻau i hoʻokahi manawa ma muli o ka pane.

Ua ʻoi aku ka maikaʻi o Macitentan a me Tadalafil ma mua o Sildenafil?

Loaʻa i nā ala lāʻau lapaʻau ʻelua ko lākou ikaika, a pili ke koho ma waena o lākou i kou kūlana olakino pilikino a me nā pahuhopu lapaʻau. Hāʻawi ka hui pū ʻana o Macitentan a me tadalafil i ka lāʻau lapaʻau ala pālua, aʻo ka sildenafil e hana ma o kahi mīkini hoʻokahi e like me ka tadalafil.

Hiki i ke ala hui pū ke hāʻawi i ka lāʻau lapaʻau piha no ka mea e kamaʻilio ana i nā ala he nui e pili ana i ka PAH. Hōʻike kekahi mau haʻawina e hiki ke ʻoi aku ka maikaʻi o ka lāʻau lapaʻau pālua ma mua o ka lāʻau lapaʻau hoʻokahi no kekahi poʻe maʻi.

Eia naʻe, ua hoʻohana ʻia ka sildenafil no ka lōʻihi no ka mālama ʻana i ka PAH a loaʻa nā ʻikepili palekana nui. Hiki ke makemake ʻia no nā poʻe maʻi e pono ai ke ala lapaʻau maʻalahi a i ʻole nā ​​kūlana olakino kūikawā e hoʻolilo i ka lāʻau lapaʻau hui ʻana i mea kūpono ʻole.

E noʻonoʻo kāu kauka i nā mea e like me ke koʻikoʻi o kou maʻi, nā kūlana olakino ʻē aʻe, nā lāʻau lapaʻau o kēia manawa, a me nā pahuhopu lapaʻau i ka wā e hoʻoholo ai i ke koho maikaʻi loa iā ʻoe.

Nā nīnau i nīnau pinepine ʻia e pili ana iā Macitentan a me Tadalafil

He palekana ʻo Macitentan a me Tadalafil no ka maʻi puʻuwai?

Hiki ke hoʻohana ʻia kēia hui pū ʻana i nā poʻe me kekahi mau ʻano o ka maʻi puʻuwai, akā pono ia i ka nānā pono ʻana a me ka loiloi ʻana e kāu kauka. No ka mea e pili ana ka PAH i ka puʻuwai, ʻo ka mālama ʻana i ke kūlana kumu e kōkua pinepine i ka hoʻomaikaʻi ʻana i ka hana o ka puʻuwai.

Eia naʻe, inā loaʻa iā ʻoe ka maʻi puʻuwai koʻikoʻi, ka puʻuwai puʻuwai hou, a i ʻole kekahi mau pilikia o ka puʻuwai, pono paha kāu kauka e hoʻoponopono i kāu hoʻolālā lapaʻau a i ʻole e noʻonoʻo i nā lāʻau lapaʻau ʻē aʻe. Hiki i ka lāʻau lapaʻau ke hoʻopilikia i ke koko a me ka helu o ka puʻuwai, no laila he mea nui ka nānā ʻana i ka puʻuwai maʻamau.

E hana pū ana kāu kauka cardiologist a me ka loea PAH e hōʻoia i ka palekana o kāu hoʻolālā lapaʻau i ka maʻi hypertension pulmonary a me nā maʻi puʻuwai e kū nei.

He aha kaʻu e hana ai inā ua hoʻohana hewa au i ka nui o Macitentan a me Tadalafil?

Inā ua lawe hewa ʻoe i ka nui o kāu lāʻau i kauoha ʻia, e kelepona koke i kāu kauka a i ʻole ke kikowaena hoʻomalu lāʻau make, ʻoiai inā maikaʻi ʻoe. Hiki i ka overdose ke hoʻoulu i ka hāʻule ʻana o ke koko a me nā pilikia koʻikoʻi.

ʻO nā hōʻailona o ka lawe ʻana i ka nui e komo paha i ka dizziness nui, ka ʻeha, ka nausea, a i ʻole nā ​​hoʻololi ʻike. Mai ho'āʻo e mālama iā ʻoe iho i kēia mau hōʻailona, ​​a mai kali e ʻike inā e hoʻomaikaʻi lākou iā lākou iho.

Ke kāhea ʻoe i ke kōkua, e loaʻa kāu ʻōmole lāʻau lapaʻau i hiki iā ʻoe ke hāʻawi i ka ʻike kikoʻī e pili ana i kāu mea i lawe ai a me ka nui. Kōkua kēia i nā poʻe loea lapaʻau e hāʻawi iā ʻoe i ka ʻōlelo aʻo kūpono loa.

He aha kaʻu e hana ai inā ua poina iaʻu kahi lāʻau o Macitentan a me Tadalafil?

Inā poina iā ʻoe kahi lāʻau, e lawe koke iā ia ke hoʻomanaʻo ʻoe, ke ʻole kokoke ka manawa no kāu lāʻau i hoʻonohonoho ʻia. I kēlā hihia, e lele i ka lāʻau i poina a hoʻomau me kāu papa hana maʻamau.

Mai lawe i ʻelua lāʻau i ka manawa hoʻokahi e hoʻoponopono ai i kahi lāʻau i poina, no ka mea, hiki i kēia ke hoʻonui i kou pilikia o nā hopena ʻaoʻao a me nā pilikia. Hiki i ka pālua-dosing ke hoʻoulu i ka hāʻule ʻana o ke koko.

Inā poina pinepine ʻoe i nā lāʻau, e noʻonoʻo e hoʻonohonoho i nā mea hoʻomanaʻo kelepona a i ʻole ka hoʻohana ʻana i kahi mea hoʻonohonoho pila e kōkua iā ʻoe e noho ma ke ala me kāu papa hana lapaʻau.

I ka manawa hea e hiki ai iaʻu ke hooki i ka lawe ʻana iā Macitentan a me Tadalafil?

Pono ʻoe e hooki i ka lawe ʻana i kēia lāʻau ma lalo o ka nānā pono ʻana a kāu kauka, no ka mea, he maʻi maʻi ʻo PAH e koi ai i ka mālama mau. ʻO ka hooki ʻana i ka hikiwawe hiki ke hoʻihoʻi a hoʻonui paha i kāu mau hōʻailona.

Hiki i kāu kauka ke noʻonoʻo e hōʻemi a i ʻole e hoʻōki i ka lāʻau lapaʻau inā loaʻa iā ʻoe nā hopena ʻaoʻao koʻikoʻi ʻaʻole hiki ke mālama ʻia, a i ʻole inā loli nui kou kūlana. Pono e hana mālie ʻia nā loli i kāu hoʻolālā lapaʻau a me ka nānā pono ʻana.

ʻOiai inā ʻoe e manaʻo maikaʻi loa, e hoʻomau i ka lawe ʻana i kāu lāʻau lapaʻau e like me ke kau ʻia. Hōʻike ka hoʻomaikaʻi ʻana i kāu mau hōʻailona e hana ana ka lāʻau lapaʻau, ʻaʻole ʻoe e pono hou.

Hiki iaʻu ke inu i ka waiʻona i ka wā e lawe ana i ka Macitentan a me Tadalafil?

Pono ʻoe e kaupalena i ka inu ʻana i ka waiʻona i ka wā e lawe ana i kēia lāʻau lapaʻau, no ka mea, hiki i ka waiʻona a me ka lāʻau lapaʻau ke hoʻohaʻahaʻa i ke koko. ʻO ka hui pū ʻana iā lākou e hoʻonui i kou pilikia o ka dizziness, fainting, a i ʻole nā hopena ʻē aʻe.

Inā koho ʻoe e inu i kekahi manawa, e hana me ka maʻalahi a e nānā i kou manaʻo. E hoʻomaka me nā mea liʻiliʻi e ʻike pehea e pane ai kou kino, a e pale i ka inu ʻana inā ʻoe e ʻike nei i ka dizziness a i ʻole ke koko haʻahaʻa.

E kamaʻilio me kāu kauka e pili ana i ke kiʻekiʻe o ka inu ʻana i ka waiʻona, inā he, palekana iā ʻoe e pili ana i kou olakino holoʻokoʻa a me ka pane ʻana i ka lāʻau lapaʻau.

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