

Health Library
October 10, 2025
Question on this topic? Get an instant answer from August.
He lāʻau lapaʻau i kuhikuhi ʻia ka Methylnaltrexone bromide i hoʻolālā ʻia e kōkua i ka mālama ʻana i ka constipation i hoʻokumu ʻia e ka opioid i nā pākeke. Inā ʻoe e lawe ana i nā lāʻau lapaʻau ʻeha opioid a ke hakakā nei me ka constipation koʻikoʻi, hana kēia lāʻau lapaʻau ma ka pale ʻana i nā mea hoʻokipa opioid i loko o kāu ʻōnaehana digestive me ka ʻole e pili ana i ka hōʻoluʻolu ʻeha. Ua hana kūikawā ʻia no ka poʻe ʻaʻole i hāʻawi nā laxatives maʻamau i ka hōʻoluʻolu kūpono mai kēia hopena ʻaoʻao paʻakikī.
Aia ka Methylnaltrexone bromide i kahi papa o nā lāʻau lapaʻau i kapa ʻia he opioid antagonists. E noʻonoʻo iā ia he mea kōkua i manaʻo ʻia e hana kūikawā i loko o kou ʻōpū digestive e kūʻē i ka constipation i hana ʻia e nā lāʻau opioid. ʻAʻole like me nā lāʻau lapaʻau constipation ʻē aʻe, ua hoʻolālā ʻia kēia lāʻau lapaʻau e hoʻoponopono i ke kumu kumu ma mua o nā hōʻailona.
Hele mai ka lāʻau lapaʻau i ke ʻano papa a lawe ʻia e ka waha. Ua hoʻomohala pono ʻia e hana kūloko i loko o kou ʻōpū me ka ʻole e hele i loko o kou lolo, ʻo ia hoʻi ʻaʻole ia e keakea i ka pono o kāu lāʻau lapaʻau ʻeha. ʻO kēia ala i manaʻo ʻia e waiwai nui ai no ka poʻe e pono ai ka lāʻau opioid e hoʻomau nei akā makemake i ka hōʻoluʻolu mai nā hopena ʻaoʻao digestive.
Hoʻohana nui ʻia kēia lāʻau lapaʻau no ka constipation i hoʻokumu ʻia e ka opioid i nā pākeke me ka ʻeha maʻi ʻole i ka maʻi maʻi. Inā ʻoe e lawe ana i nā lāʻau lapaʻau ʻeha opioid e like me ka morphine, oxycodone, a i ʻole fentanyl no ka manawa lōʻihi, hiki iā ʻoe ke ʻike i ka constipation koʻikoʻi ʻaʻole e pane maikaʻi i nā laxatives kuʻuna.
Hiki i kāu kauka ke ʻōlelo aku i ka methylnaltrexone bromide inā ua hoʻāʻo ʻoe i nā lāʻau lapaʻau ʻē aʻe no ka paʻa ʻana o ka ʻōpū me ka holopono ʻole. Ua hoʻolālā ʻia ka lāʻau lapaʻau no nā kūlana kahi e pono ai nā lāʻau opioid, akā ʻo ka paʻa ʻana o ka ʻōpū e hana ai e hoʻopilikia nui i kou ola. ʻAʻole ia i manaʻo ʻia no ka paʻa ʻana o ka ʻōpū i kekahi manawa a i ʻole ka paʻa ʻana o ka ʻōpū mai nā kumu ʻē aʻe.
Hana ka methylnaltrexone bromide ma ka pale ʻana i nā mea loaʻa opioid i loko o kāu ʻōnaehana digestive. Ke lawe ʻoe i nā lāʻau lapaʻau ʻeha opioid, pili lākou i nā mea loaʻa ma kou kino a pau, me kou ʻōpū, e lohi ai i nā neʻe ʻana o ka ʻōpū a hoʻoulu i ka paʻa ʻana o ka ʻōpū.
Hana kēia lāʻau lapaʻau e like me ka mea pale koho e pale ai i nā opioids mai ka pili ʻana i nā mea loaʻa i loko o kou ʻōpū. ʻO ka mea nui, ʻaʻole ia e hele i ka pale koko-lolo, no laila ʻaʻole ia e hōʻemi i ka pono o kāu lāʻau lapaʻau ʻeha. Manaʻo ʻia he lāʻau lapaʻau ikaika waena e hana pono ana i kahi e pono ai.
Hoʻomaka ka hapa nui o nā kānaka e ʻike i nā hopena i loko o kekahi mau hola a i ʻole i ka lā ma hope o ka lawe ʻana i ka lāʻau lapaʻau. He mea maʻamau ka hopena akā mālie, e kōkua ana i ka hoʻihoʻi ʻana i ka hana ʻōpū maʻamau me ka ʻole e hana i ka wikiwiki a i ʻole ka hōʻoluʻolu ʻole.
E lawe i ka methylnaltrexone bromide e like me ke kauoha a kāu kauka, maʻamau hoʻokahi manawa i ka lā ma ka ʻōpū ʻole. Hana maikaʻi ka lāʻau lapaʻau ke lawe ʻia ma kahi o 30 mau minuke ma mua o kāu ʻai mua o ka lā a i ʻole ma kahi o ʻelua hola ma hope o ka ʻai ʻana.
E ale i ka papa holoʻokoʻa me ke aniani wai piha. Mai ʻoki, nau, a i ʻole e wāwahi i ka papa, no ka mea, hiki i kēia ke hoʻopilikia i ke ʻano o ka lawe ʻia ʻana a me ka hoʻokuʻu ʻia ʻana o ka lāʻau lapaʻau i loko o kou kino. Inā pilikia ʻoe i ka ale ʻana i nā pila, e kamaʻilio me kāu kauka e pili ana i nā koho ʻē aʻe ma mua o ka hoʻololi ʻana i ka papa.
E hoʻāʻo e lawe i kāu lāʻau i ka manawa like i kēlā me kēia lā e mālama i nā pae kūlike i loko o kou kino. Inā ʻoe e ʻai i ka meaʻai momona nui, hiki iā ia ke hōʻemi i ka pono o ka lāʻau, no laila he mea nui ka manawa e pili ana i nā meaʻai no nā hopena maikaʻi loa.
Aia ka lōʻihi o ka mālama ʻana i ka lōʻihi o kou pono i ka lāʻau ʻeha opioid. No ka mea ua hoʻolālā ʻia ka methylnaltrexone bromide e kūʻē i ka constipation i hoʻokumu ʻia e ka opioid, e hoʻomau paha ʻoe i ka lawe ʻana iā ia i ka wā e mālama ʻia ai ʻoe i ka opioid a me ka ʻike ʻana i ka constipation.
E loiloi mau kāu kauka inā pono a pono ka lāʻau lapaʻau no kou kūlana. Pono paha kekahi poʻe i nā pule a i ʻole nā mahina, ʻoiai e pono ana kekahi i ka mālama lōʻihi. ʻO ke kī ka loaʻa ʻana o ke kaulike kūpono ma waena o ka mālama ʻana i kou ʻeha a me ka mālama ʻana i ka hana ʻōpū ʻoluʻolu.
Mai hooki koke i ka lawe ʻana i kēia lāʻau me ka ʻole e kūkākūkā i kāu kauka, ʻoiai inā e lawe ana ʻoe i nā lāʻau ʻeha opioid. E kōkua kāu mea mālama ola iā ʻoe e hoʻoholo i ka lōʻihi o ka mālama kūpono e pili ana i kāu mau pono pilikino a me ka pane ʻana i ka lāʻau.
E like me nā lāʻau lapaʻau a pau, hiki i ka methylnaltrexone bromide ke hana i nā hopena ʻaoʻao, ʻoiai ʻaʻole ʻike nā mea a pau iā lākou. ʻO ka hoʻomaopopo ʻana i ka mea e manaʻo ai hiki ke kōkua iā ʻoe e mākaukau a ʻike i ka manawa e hoʻopili ai i kāu mea mālama ola.
ʻO nā hopena ʻaoʻao maʻamau e ʻike ai ka poʻe he nui:
He maʻalahi kēia mau hopena a maʻa mau e hoʻomaikaʻi i ka wā e hoʻoponopono ai kou kino i ka lāʻau. ʻIke ka hapa nui o ka poʻe i ka hoʻomaka ʻana me ka lāʻau haʻahaʻa loa e kōkua i ka hōʻemi ʻana i kēia mau hopena ʻaoʻao mua.
ʻO nā hopena ʻaoʻao liʻiliʻi akā ʻoi aku ka koʻikoʻi e koi ai i ka lāʻau lapaʻau koke:
I nā manawa kakaʻikahi, hiki i kekahi poʻe ke loaʻa nā hopena maʻi a i ʻole ka puka ʻana o ka ʻōpū. Inā ʻoe e ʻike i ka ʻeha nui o ka ʻōpū, ke kuni, a i ʻole nā hōʻailona o ka hopena maʻi e like me ka ʻūhū a i ʻole ka pilikia o ka hanu ʻana, e ʻimi koke i ka lāʻau lapaʻau ulia pōpilikia.
Pono kekahi poʻe e pale i ka methylnaltrexone bromide ma muli o nā pilikia palekana. E nānā pono kāu kauka i kāu mōʻaukala olakino ma mua o ke kau ʻana i kēia lāʻau lapaʻau e hōʻoia i ka kūpono no kou kūlana.
ʻAʻole pono ʻoe e lawe i kēia lāʻau lapaʻau inā loaʻa iā ʻoe:
Pono ka poʻe me kekahi mau maʻi i ka mālama hou a me ka nānā pono ʻana. E kaupaona kāu kauka i nā pōmaikaʻi a me nā pilikia inā loaʻa iā ʻoe ka mōʻaukala o ke ʻoki ʻana i ka ʻōpū, ka maʻi o Crohn, a i ʻole nā maʻi ʻē aʻe o ka ʻōpū.
Pono nā wahine hāpai a me nā wahine e hānai ana i ka waiū e kūkākūkā i nā pilikia a me nā pōmaikaʻi me kā lākou mea mālama ola, no ka mea, ʻaʻole i hoʻokumu ʻia ka palekana o kēia lāʻau lapaʻau i ka wā o ka hāpai ʻana a me ka lactation.
Loaʻa ka methylnaltrexone bromide ma lalo o ka inoa inoa Relistor. Hana ʻia kēia inoa e Bausch Health a ʻo ia ke ʻano i kauoha pinepine ʻia o kēia lāʻau lapaʻau ma ʻAmelika Hui Pū ʻIa.
Hiki nō hoʻi iā ʻoe ke loaʻa nā mana generic o ka methylnaltrexone bromide, aia i loko o ka mea hana like akā ʻoi aku ka maʻalahi. Pono nā lāʻau lapaʻau generic e hoʻokō i nā kūlana palekana a me ka pono like me nā lāʻau lapaʻau inoa inoa, no laila he mau koho hilinaʻi like lākou.
E nānā mau me kāu mea kūʻai lāʻau lapaʻau inā ʻoe e hoʻololi ana ma waena o nā mana brand a me nā mana generic, no ka mea, aia paha nā ʻokoʻa liʻiliʻi i nā mea hana ʻole e pili ana i ke ʻano o kou ʻae ʻana i ka lāʻau.
Nui nā lāʻau lapaʻau ʻē aʻe e hiki ke kōkua i ka mālama ʻana i ka constipation i hoʻokumu ʻia e ka opioid inā ʻaʻole kūpono ka methylnaltrexone bromide iā ʻoe. Hana ʻokoʻa kēlā me kēia koho a ʻoi aku paha ka maikaʻi no kāu kūlana kikoʻī a me ka mōʻaukala olakino.
ʻO nā mea kūʻē opioid ʻē aʻe e komo pū ana me naloxegol (Movantik) a me naldemedine (Symproic). Hana like kēia mau lāʻau lapaʻau me methylnaltrexone bromide ma ka pale ʻana i nā mea hoʻokipa opioid i loko o ka ʻōnaehana digestive me ka mālama ʻana i ka hōʻoluʻolu ʻeha.
Hiki nō hoʻi i nā laxatives kuʻuna e like me docusate, senna, a i ʻole polyethylene glycol ke kōkua, ʻoi aku ka nui ke hoʻohana ʻia i ka hui pū ʻana. Loaʻa i kekahi poʻe ka holomua me nā ala ola e like me ka hoʻonui ʻana i ka wai, ka fiber meaʻai, a me ka hoʻoikaika kino mālie, ʻoiai ʻaʻole lawa paha kēia mau ʻano hana no ka constipation i hoʻokumu ʻia e ka opioid.
Hiki i kāu kauka ke kōkua iā ʻoe e ʻimi i kēia mau koho ʻē aʻe a hoʻoholo i ke ala a i ʻole ka hui pū ʻana o nā lāʻau lapaʻau e hana maikaʻi loa no kāu mau pono pilikino.
He mau lāʻau lapaʻau maikaʻi ʻo Methylnaltrexone bromide a me naloxegol (Movantik) no ka constipation i hoʻokumu ʻia e ka opioid, akā he mau ʻokoʻa nui ko lākou. ʻO ke koho ma waena o lākou e hilinaʻi pinepine ʻia i kāu mau makemake pilikino, ka mōʻaukala olakino, a me ka maikaʻi o kou ʻae ʻana i kēlā me kēia lāʻau.
Lawe ʻia ka Methylnaltrexone bromide i hoʻokahi manawa i ka lā a hiki ke hana wikiwiki iki no kekahi poʻe, e hāʻawi pinepine ana i ka hōʻoluʻolu i loko o nā hola. Lawe ʻia ʻo Naloxegol i hoʻokahi manawa i ka lā akā loaʻa paha kahi hana mālie, kahi e makemake ai kekahi poʻe.
Ma ke ʻano o nā hopena ʻē aʻe, hiki i nā lāʻau lapaʻau ʻelua ke hana i nā hōʻailona digestive like e like me ka ʻeha o ka ʻōpū a me ka maʻi maʻi. Eia naʻe, ʻokoʻa loa ka ʻae ʻana o kēlā me kēia kanaka, a ʻo ka mea e hana maikaʻi ai no kekahi kanaka ʻaʻole paha ia he mea kūpono no kekahi.
E noʻonoʻo kāu kauka i nā mea e like me kāu mau lāʻau lapaʻau ʻē aʻe, ka hana o ka puʻupaʻa, a me nā makemake pilikino i ke kōkua ʻana iā ʻoe e koho ma waena o kēia mau koho. Ua manaʻo ʻia lāua ʻelua he mau lāʻau lapaʻau mua no ka constipation i hoʻokumu ʻia e ka opioid.
Ua manaʻo ʻia ʻo Methylnaltrexone bromide he palekana no ka poʻe me ka maʻi puʻuwai, akā pono kāu kauka e loiloi i kou kūlana cardiac kikoʻī. ʻAʻole pili pololei ka lāʻau lapaʻau i ka hana o ka puʻuwai, akā pono e nānā ʻia nā loli i kou olakino holoʻokoʻa.
Inā loaʻa iā ʻoe ka maʻi puʻuwai koʻikoʻi a i ʻole e lawe i nā lāʻau lapaʻau cardiac he nui, makemake paha kāu kauka e hoʻomaka me ka haʻahaʻa haʻahaʻa a nānā pono iā ʻoe. ʻO ke kī, ʻo ia ka hōʻoia ʻana ʻaʻole e hoʻopilikia nā hopena ʻē aʻe i ka ʻai ʻana i kāu lāʻau lapaʻau puʻuwai a i ʻole ke kūpaʻa cardiovascular holoʻokoʻa.
Inā lawe hewa ʻoe i ka nui o kāu kauoha, e hoʻokaʻaʻike koke i kāu kauka a i ʻole ke kikowaena mana ʻawaʻawa. ʻO ka lawe ʻana i ka nui o ka methylnaltrexone bromide hiki ke alakaʻi i ka maʻi maʻi koʻikoʻi, ka dehydration, a me nā kaulike electrolyte e pono ai ka lāʻau lapaʻau.
Mai ho'āʻo e pale i ka overdose ma ka lawe ʻana i nā lāʻau lapaʻau ʻē aʻe a i ʻole ke kāpae ʻana i kāu lāʻau lapaʻau ʻeha opioid. Akā, e kālele ana i ka noho ʻana i ka wai a me ka ʻimi ʻana i ke alakaʻi lapaʻau ʻoihana. E mālama i ka hue lāʻau me ʻoe i ka wā e ʻimi ai i ke kōkua i hiki i nā mea mālama ola ke ʻike pololei i ka mea a me ka nui āu i lawe ai.
Inā ʻoe e poina i kahi lāʻau, e lawe koke iā ia ke hoʻomanaʻo ʻoe, inā aia nō ia ma ka ʻōpū ʻole. Inā kokoke i kāu lāʻau i hoʻonohonoho ʻia e hiki mai ana a i ʻole ua ʻai ʻoe i kēia manawa, e lele i ka lāʻau i poina a e hoʻomau me kāu papa manawa maʻamau.
Mai lawe i ʻelua lāʻau i ka manawa hoʻokahi e uku ai i kahi lāʻau i poina, no ka mea, hiki i kēia ke hoʻonui i kou pilikia o nā hopena ʻaoʻao. Ma kahi o ia mea, e hoʻi i kāu papa manawa maʻamau a e hoʻokaʻaʻike i kāu kauka inā he nīnau kāu e pili ana i ka mālama ʻana i nā lāʻau i poina.
Hiki iā ʻoe ke hooki i ka lawe ʻana i ka methylnaltrexone bromide ke pono ʻole ʻoe i ka lāʻau ʻeha opioid a i ʻole ke hoʻoponopono ʻia kou paʻa ʻana. Eia naʻe, he mea nui e kūkākūkā i kēia hoʻoholo me kāu kauka ma mua o ka hooki ʻana me ka wikiwiki.
E kōkua kāu mea mālama ola iā ʻoe e hoʻoholo i ka manawa kūpono e hooki ai i ka lāʻau lapaʻau e pili ana i kāu mau pono mālama ʻeha a me nā hōʻailona digestive. Pono paha kekahi poʻe e hoʻemi mālie, a hiki i nā poʻe ʻē aʻe ke hooki koke me ka pilikia ʻole.
Ma keʻano maʻamau, pono ʻoe e pale i ka lawe ʻana i nā laxatives ʻē aʻe i ka wā e hoʻohana ana i ka methylnaltrexone bromide ke ʻole i kuhikuhi ʻia e kāu kauka. ʻO ka hui ʻana i nā lāʻau lapaʻau paʻa he nui hiki ke alakaʻi i nā hopena hiki ʻole ke wānana a hiki ke hana i ka maʻi palahī a i ʻole ka maloʻo.
Inā manaʻo ʻoe ʻaʻole hāʻawi wale ka methylnaltrexone bromide i ka hoʻomaha kūpono, e kamaʻilio me kāu mea mālama ola e pili ana i ka hoʻoponopono ʻana i kāu hoʻolālā lapaʻau. Hiki iā lākou ke ʻōlelo e hoʻololi i kāu lāʻau, e hoʻololi i nā lāʻau lapaʻau, a i ʻole e kamaʻilio i nā mea ʻē aʻe e hiki ke kōkua i kou paʻa ʻana.
6Mpeople
Get clear medical guidance
on symptoms, medications, and lab reports.