

Health Library
October 10, 2025
Question on this topic? Get an instant answer from August.
He lāʻau lapaʻau i kauoha ʻia ka Methylnaltrexone e kōkua i ka hoʻomaha ʻana i ka paʻa ʻana o ka ʻōpū i hana ʻia e nā lāʻau ʻeha opioid. Inā ʻoe e lawe ana i nā opioids no ka mālama ʻeha a e hakakā nei me ka paʻa ʻana o ka ʻōpū, hiki i kēia lāʻau lapaʻau ke hāʻawi i ke kōkua me ka ʻole e hoʻopilikia i kāu kaohi ʻeha. Hana ia ma ka pale ʻana i nā hopena opioid ma kāu ʻōnaehana digestive me ka waiho ʻana i ka hoʻomaha ʻeha i ka wā o ke kino.
He lāʻau lapaʻau kūikawā ka Methylnaltrexone i hoʻolālā ʻia e mālama i ka paʻa ʻana o ka ʻōpū i hoʻokumu ʻia e ka opioid. No ka papa o nā lāʻau i kapa ʻia he opioid antagonists, ʻo ia hoʻi, e pale ana i kekahi mau hopena opioid i nā ʻāpana kikoʻī o kou kino. Hele mai ka lāʻau lapaʻau ma ke ʻano he subcutaneous injection, ʻo ia hoʻi, hāʻawi ʻia ma ke ʻano he pana ma lalo o kou ʻili, e like me ke ʻano o ka poʻe me ka maʻi diabetes e hāʻawi iā lākou iho i nā injections insulin.
Ua hana kūikawā ʻia kēia lāʻau lapaʻau e hana wale i kāu ʻōnaehana digestive a ʻaʻole e hele i loko o kou lolo. ʻO kēia hoʻolālā kūʻokoʻa ʻo ia ke hiki ke hoʻihoʻi i ka hana ʻōpū maʻamau me ka ʻole e hōʻemi i ka hoʻomaha ʻeha āu e loaʻa ai mai kāu mau lāʻau opioid. He mea kōkua nui ia no ka poʻe e pono ai ka lāʻau lapaʻau opioid lōʻihi akā ke ʻike nei i ka paʻa ʻana o ka ʻōpū ma ke ʻano he hopena ʻaoʻao.
Hoʻomaʻamaʻa ʻo Methylnaltrexone i ka paʻa ʻana o ka ʻōpū i hoʻokumu ʻia e ka opioid i nā pākeke e lawe mau ana i nā lāʻau ʻeha opioid. He ʻokoʻa kēia ʻano paʻa ʻana o ka ʻōpū mai ka paʻa ʻana o ka ʻōpū maʻamau no ka mea ua hana ʻia e nā opioids e hoʻolohi ana i kāu ʻōnaehana digestive. Nui ka poʻe e lawe ana i nā opioids no ka ʻeha mau, ka maʻi maʻi, a i ʻole ma hope o ke ʻoki ʻana e ʻike i kēia hopena ʻaoʻao paʻakikī.
Hoʻohana ʻia ka lāʻau lapaʻau i ka wā i hana ʻole ai nā lāʻau lapaʻau ʻē aʻe no ka paʻa ʻana o ka ʻōpū. Hiki i kāu kauka ke ʻōlelo aku iā ia inā ua hoʻāʻo ʻoe i ka fiber i hoʻonui ʻia, nā mea palupalu o ka noho, a i ʻole nā laxatives me ka ʻole o ka hōʻoluʻolu kūpono. He mea waiwai loa ia no ka poʻe e pono e hoʻomau i ka lawe ʻana i nā opioids no ka mālama ʻana i ka ʻeha akā makemake e hoʻihoʻi i ka hana ʻōpū maʻamau.
I kekahi mau hihia, kuhikuhi nā kauka i ka methylnaltrexone no ka poʻe me ka maʻi holomua e loaʻa ana i ka mālama palliative. Kōkua kēia i ka hoʻomaikaʻi ʻana i ka maikaʻi o ke ola ma ka hoʻoponopono ʻana i kekahi o nā hopena ʻaoʻao ʻoluʻolu ʻole o ka lāʻau lapaʻau ʻeha.
Hana ʻo Methylnaltrexone ma ka pale ʻana i nā mea hoʻokipa opioid ma kāu ʻōnaehana digestive. Ke lawe ʻoe i nā lāʻau lapaʻau ʻeha opioid, pili lākou i nā mea hoʻokipa ma kou kino, me kou ʻōpū. ʻOiai hāʻawi kēia i ka hōʻoluʻolu ʻeha, hoʻolohi pū ia i ka neʻe ʻana o ka meaʻai a me ka ʻōpala ma kou ʻōnaehana digestive, e alakaʻi ana i ka paʻa ʻana o ka ʻōpū.
Hoʻolālā ʻia kēia lāʻau lapaʻau me kahi ʻano kūikawā e pale ai i ka hele ʻana i ka pale koko-lolo. ʻO ia hoʻi, ʻaʻole hiki iā ia ke hiki i nā mea hoʻokipa opioid i kou lolo e kāohi i ka hōʻoluʻolu ʻeha. Akā, e kālele ana ia i nā mea hoʻokipa opioid i loko o kou ʻōpū, e ʻae ana i kāu ʻōnaehana digestive e hana maʻamau me ka mālama ʻana i kāu lāʻau lapaʻau ʻeha.
Manaʻo ʻia ka lāʻau lapaʻau he ikaika a hana maʻamau i ka neʻe ʻana o ka ʻōpū i loko o kekahi mau hola i ka lā ma hope o ka injection. ʻIke ka hapa nui o ka poʻe he mea maikaʻi loa ia no kāna kumu i manaʻo ʻia, ʻoiai hiki ke ʻokoʻa nā pane pilikino ma muli o nā mea e like me kou olakino holoʻokoʻa a me ka lōʻihi o kou lawe ʻana i nā opioids.
Hāʻawi ʻia ka methylnaltrexone ma ke ʻano he injection subcutaneous, ʻo ia hoʻi e hoʻokomo ʻoe a i ʻole kekahi mea mālama iā ia ma lalo o ka ʻili. E aʻo kāu mea mālama ola iā ʻoe i ke ʻano hoʻokomo kūpono a hōʻike iā ʻoe i nā wahi hoʻokomo maikaʻi loa, maʻamau kou ʻūhā, ʻōpū, a i ʻole ka lima luna. Hāʻawi ʻia ka injection i kēlā me kēia lā ʻē aʻe, akā e hoʻoholo kāu kauka i ka papa manawa kūpono no kou kūlana.
ʻAʻole pono ʻoe e lawe i kēia lāʻau me ka meaʻai, a ʻaʻohe palena meaʻai kikoʻī. Eia naʻe, he mea nui e noho maikaʻi i ka wai ke hoʻohana ʻoe i kekahi lāʻau e pili ana i ka hana ʻōpū. Pono e hāʻawi ʻia ka injection ma ka lumi wela, no laila pono ʻoe e wehe iā ia mai ka pahu hau ma kahi o 30 mau minuke ma mua o ka hoʻokomo ʻana.
E hoʻololi mau i kāu mau wahi injection e pale ai i ka huhū o ka ʻili a i ʻole ka pōʻino o ka ʻiʻo. E mālama i kahi āu i hoʻokomo ai i kēia manawa a koho i kahi ʻokoʻa i kēlā me kēia manawa. Inā ʻoluʻolu ʻole ʻoe i ka hāʻawi ʻana iā ʻoe iho i nā injections, hiki i kahi lālā o ka ʻohana a i ʻole ka mea mālama ke aʻo e kōkua iā ʻoe, a i ʻole hiki iā ʻoe ke loaʻa nā injections ma ke keʻena o kāu kauka.
Aia ka lōʻihi o ka mālama ʻana i ka methylnaltrexone i ka lōʻihi o kou pono e lawe i nā lāʻau lapaʻau ʻeha opioid. No ka mea e mālama ana kēia lāʻau i kahi hopena ʻaoʻao o nā opioids ma mua o kahi maʻi maʻi, e hoʻohana maʻamau ʻoe iā ia no ka lōʻihi o kou ʻike ʻana i ka constipation i hoʻokomo ʻia e ka opioid. Hiki paha kēia i nā pule, nā mahina, a i ʻole ka lōʻihi no ka poʻe me nā maʻi ʻeha mau.
E loiloi mau kāu kauka inā pono ʻoe i ka lāʻau. Inā emi kāu ʻano opioid a i ʻole inā e hooki ʻoe i ka lawe ʻana i nā opioids, e hiki nō paha iā ʻoe ke hoʻōki i ka methylnaltrexone. ʻIke kekahi poʻe e hoʻomaikaʻi ana ko lākou constipation i hiki iā lākou ke hoʻokele me nā lāʻau lapaʻau ʻē aʻe, e ʻae iā lākou e hoʻōki i nā injections.
He mea nui ʻaʻole e hooki koke i ka methylnaltrexone me ke kamaʻilio ʻole ʻana me kāu mea mālama ola. ʻOiai ʻaʻole ia he mea e hana ai i ka maʻamau, ʻo ka hooki koke ʻana e hoʻi koke mai paha kou paʻa ʻana. Hiki i kāu kauka ke kōkua iā ʻoe e hoʻoholo i ke ala maikaʻi loa no kou kūlana.
Hoʻomanawanui ka hapa nui o nā kānaka i ka methylnaltrexone, akā e like me nā lāʻau lapaʻau a pau, hiki iā ia ke hana i nā hopena ʻaoʻao. ʻO nā hopena ʻaoʻao maʻamau he maʻalahi a pili i nā loli i kāu ʻōnaehana digestive i ka wā e hoʻoponopono ai i ka hana maʻamau.
Eia nā hopena ʻaoʻao maʻamau e hiki iā ʻoe ke ʻike:
Hoʻomaikaʻi pinepine kēia mau hopena ʻaoʻao maʻamau i ka wā e hoʻoponopono ai kou kino i ka lāʻau a me ka hoʻopaʻa ʻana o kāu hana ʻōpū.
Aia kekahi mau hopena ʻaoʻao liʻiliʻi akā ʻoi aku ka koʻikoʻi e ʻike ai:
Inā loaʻa iā ʻoe kekahi mau hōʻailona koʻikoʻi a i ʻole nā mea e hopohopo ai, e kelepona koke i kāu mea mālama ola. ʻO ka hapa nui o nā kānaka e ʻike i nā pōmaikaʻi o ka hana ʻana o ka ʻōpū i ʻoi aku ka maikaʻi ma mua o ka hōʻoluʻolu manawa o nā hopena ʻaoʻao.
ʻAʻole palekana ʻo Methylnaltrexone no nā mea a pau, a aia kekahi mau kūlana koʻikoʻi kahi e pono ʻole ai e hoʻohana ʻia. E nānā pono kāu kauka i kāu moʻolelo olakino ma mua o ka kau ʻana i kēia lāʻau lapaʻau e hōʻoia i ka palekana iā ʻoe.
ʻAʻole pono ʻoe e lawe i ka methylnaltrexone inā loaʻa iā ʻoe kekahi o kēia mau kūlana:
E hoʻohana pū kāu kauka i ka mālama keu inā loaʻa iā ʻoe kekahi mau kūlana ʻē aʻe e hiki ke hoʻonui i kou pilikia o nā pilikia:
E haʻi mau i kāu mea mālama ola e pili ana i kāu mau maʻi olakino a me nā lāʻau lapaʻau i kēia manawa ma mua o ka hoʻomaka ʻana i ka methylnaltrexone. Kōkua kēia i ka hōʻoia ʻana i ka palekana a me ka maikaʻi o ka lāʻau lapaʻau no kāu kūlana.
Loaʻa ʻo Methylnaltrexone ma lalo o ka inoa inoa Relistor. ʻO kēia ke ʻano i kuhikuhi pinepine ʻia o ka lāʻau lapaʻau a hele mai i nā syringes i hoʻopiha mua ʻia no ka injection subcutaneous. Loaʻa i ka mana inoa inoa a me nā mana generic i ka mea hana like a hana like.
Hiki i kekahi mau hoʻolālā ʻinikua ke makemake i ka inoa inoa versus nā lāʻau lapaʻau generic, no laila pono e nānā me kāu mea hoʻolako ʻinikua e pili ana i ka uhi. Hiki i kāu kauka lapaʻau ke kōkua iā ʻoe e hoʻomaopopo i kāu mau koho a me nā ʻokoʻa kumukūʻai ma waena o nā formulations i loaʻa.
Inā ʻaʻole kūpono ʻo methylnaltrexone iā ʻoe, aia kekahi mau koho lapaʻau ʻē aʻe no ka constipation i hoʻokomo ʻia e ka opioid. Hiki i kāu kauka ke ʻōlelo aku e hoʻāʻo i kēia mau koho ʻē aʻe e pili ana i kāu kūlana kikoʻī a me ka mōʻaukala olakino.
ʻO nā lāʻau lapaʻau ʻē aʻe no ka constipation i hoʻokomo ʻia e ka opioid:
ʻO nā ala hana ʻole i kāu kauka e ʻōlelo ai:
ʻO ke ala maikaʻi loa e pili ana i ka hui ʻana i nā hoʻolālā like ʻole. Hiki i kāu mea mālama ola ke kōkua iā ʻoe e hoʻomohala i kahi hoʻolālā piha e pili ana i kou constipation i ka wā e mālama ana i ka mana ʻeha maikaʻi.
He kūpono ʻo methylnaltrexone a me naloxegol no ka mālama ʻana i ka paʻa ʻana o ka ʻōpū i hoʻokumu ʻia e ka opioid, akā he mau pōmaikaʻi like ʻole ko lākou e pili ana i kou kūlana. ʻO ka koho ma waena o lākou e pili pinepine ana i kāu makemake, ke ʻano o ke ola, a me ke ʻano o kou kino e pane ai i kēlā me kēia lāʻau.
He ʻoi aku ka maikaʻi o Methylnaltrexone inā makemake ʻoe i ka liʻiliʻi o ka hoʻohana ʻana, no ka mea, hāʻawi ʻia ia i kēlā me kēia lā ʻē aʻe ma mua o kēlā me kēia lā. Manaʻo kekahi poʻe e hana wikiwiki a hilinaʻi ka injection ma mua o nā lāʻau lapaʻau waha. He koho maikaʻi paha ia inā pilikia ʻoe i ka hoʻomanaʻo ʻana e lawe i nā lāʻau lapaʻau i kēlā me kēia lā a i ʻole inā he pilikia digestive kou e hoʻopilikia ai i ka lawe ʻana i ka pila.
He mea makemake ʻia paha ʻo Naloxegol inā ʻaʻole ʻoluʻolu ʻoe i nā injections a i ʻole makemake ʻoe i ka maʻalahi o ka lawe ʻana i ka pila. Lawe ʻia ia i hoʻokahi manawa i ka lā ma ka waha a ʻaʻole pono i nā lako a i ʻole nā ʻenehana injection. Manaʻo kekahi poʻe he maʻalahi nā lāʻau lapaʻau waha e hoʻohui i kā lākou hana maʻamau i kēlā me kēia lā.
Hana nā lāʻau lapaʻau ʻelua ma o nā ʻano hana like a loaʻa ka pono like no ka hapa nui o nā kānaka. Hiki i kāu kauka ke kōkua iā ʻoe e kaupaona i nā mea maikaʻi a me nā mea maikaʻi ʻole o kēlā me kēia koho e pili ana i kāu mau pono pilikino, nā makemake, a me ka mōʻaukala olakino.
Pono ʻo Methylnaltrexone i ka noʻonoʻo pono inā loaʻa iā ʻoe ka maʻi kīkī. No ka mea, kōkua kou mau kīkī i ka hana ʻana a me ka hoʻopau ʻana i kēia lāʻau lapaʻau mai kou kino, hiki i nā pilikia kīkī ke hoʻopilikia i ke ʻano o ka hana ʻana o ka lāʻau a hiki ke hoʻonui i kou pilikia o nā hopena ʻaoʻao.
Inā loaʻa iā ʻoe ka maʻi kīkī māmā a i ʻole ka maʻi kīkī, hiki i kāu kauka ke kuhikuhi i kahi haʻahaʻa haʻahaʻa a i ʻole e nānā pono iā ʻoe i ka wā e lawe ana ʻoe i ka lāʻau. No ka poʻe me ka maʻi kīkī koʻikoʻi, ʻaʻole ʻōlelo ʻia ʻo methylnaltrexone no ka mea hiki ke kūkulu i loko o kāu ʻōnaehana a hoʻopilikia.
E hōʻike mau i kāu mea mālama ola e pili ana i nā pilikia kīkī āu, ʻoiai inā he mea liʻiliʻi lākou. Hiki iā lākou ke makemake e nānā i kāu hana kīkī me nā hoʻokolohua koko ma mua o ka hoʻomaka ʻana i ka lāʻau a me kēlā me kēia manawa ke lawe nei ʻoe.
Inā ua hoʻokomo hewa ʻoe i ka methylnaltrexone nui loa, e hoʻokaʻaʻike koke i kāu mea mālama ola a i ʻole ke kikowaena hoʻomalu lāʻau make. ʻOiai ʻaʻole maʻamau nā overdoses me kēia lāʻau, hiki i ka lawe ʻana i ka nui loa ke kumu i ka ʻeha nui o ka ʻōpū, ka maʻi palahī, ka nausea, a i ʻole ka luaʻi.
Mai hoʻāʻo e mālama i kahi overdose iā ʻoe iho a i ʻole e kali e ʻike inā e ulu nā hōʻailona. ʻOiai inā maikaʻi ʻoe i ka wā mua, he mea nui e kiʻi i ka ʻōlelo aʻoaʻo lapaʻau me ka wikiwiki. ʻAʻole paha e ʻike koke ʻia nā hopena o ka lāʻau nui loa akā hiki ke lilo i mea koʻikoʻi.
E mālama i ka pūʻolo lāʻau me ʻoe ke ʻimi ʻoe i ke kōkua, no ka mea, hiki i kēia ʻike ke waiwai i nā mea mālama ola. I ka wā e hiki mai ana, e nānā pālua i kāu mahele a me ke ʻano o ka hoʻokomo ʻana e pale ai i nā overdoses ulia.
Inā ua hala ʻoe i kahi mahele o methylnaltrexone, e lawe iā ia i ka wā e hoʻomanaʻo ai ʻoe, ke ʻole ua kokoke ka manawa no kāu mahele i hoʻonohonoho ʻia. I kēlā hihia, e lele i ka mahele i hala a e hoʻomau me kāu papa hana maʻamau. Mai lawe i ʻelua mahele i ka manawa hoʻokahi e hoʻoponopono ai i kahi mahele i hala.
ʻAʻole pilikia ka hala ʻana i kahi mahele i kekahi manawa, akā e ʻike paha ʻoe e hoʻi ana a ʻoi aku paha ka paʻa ʻana o kou ʻōpū no ka manawa pōkole. Inā poina pinepine ʻoe i nā mahele, e noʻonoʻo e hoʻonohonoho i nā mea hoʻomanaʻo kelepona a i ʻole e hoʻohana i kahi polokalamu mālama lāʻau e kōkua iā ʻoe e noho ma ka papa hana.
Inā hala ʻoe i nā mahele maʻamau, e kamaʻilio me kāu mea mālama ola e pili ana i nā hoʻolālā e hoʻomaikaʻi ai i ka pili ʻana a i ʻole inā he papa hana lāʻau ʻokoʻa paha e hana maikaʻi no kou ola.
Hiki iā ʻoe ke hooki i ka lawe ʻana i ka methylnaltrexone ke ʻaʻole ʻoe e pono hou ia mea no ka paʻa ʻana o ka ʻōpū i hoʻokumu ʻia e ka opioid. Hana maʻamau kēia ke hōʻemi nui ʻoe i kāu mahele opioid, hooki loa i ka lawe ʻana i nā opioids, a i ʻole e ʻike ʻoe ua hoʻomaikaʻi ʻia kou paʻa ʻana o ka ʻōpū e lawa ai e mālama me nā lāʻau lapaʻau ʻē aʻe.
E kūkākūkā mau i ka hooki ʻana i ka lāʻau lapaʻau me kāu mea mālama ola ma mua o ka hoʻoholo ʻana iā ʻoe iho. Hiki iā lākou ke kōkua iā ʻoe e hoʻoholo i ka manawa maikaʻi loa a inā pono ʻoe e hoʻemi mālie i ka mahele a i ʻole hiki ke hooki koke.
ʻIke kekahi poʻe e hoʻomaikaʻi mau ana kā lākou hana ʻōpū ʻoiai ma hope o ka hooki ʻana i ka methylnaltrexone, ʻoiai inā ua hana lākou i nā loli meaʻai a i ʻole ke ola. Pono paha kekahi poʻe e hoʻomau i ka lāʻau lapaʻau inā hoʻi ka paʻa ʻana o ka ʻōpū ke hooki lākou.
Hiki iā ʻoe ke lawe pinepine i ka methylnaltrexone me nā laxatives ʻē aʻe, akā pono e hana ʻia kēia ma lalo o ka mālama ʻana i ka lāʻau lapaʻau. Hiki i kāu kauka ke ʻōlelo e hui pū i nā lāʻau lapaʻau inā pono ʻoe i ke kōkua hou me ka paʻa ʻana o ka ʻōpū, akā makemake lākou e nānā pono iā ʻoe e pale i ka hana ʻōpū nui.
Inā ʻoe e lawe nei i nā laxatives ʻē aʻe ke hoʻomaka ʻoe i ka methylnaltrexone, hiki i kāu kauka ke hoʻoponopono i kēlā mau mahele e pale i ka maʻi maʻi a i ʻole ka ʻeha. Hiki i ka hui pū ʻana o nā lāʻau lapaʻau ke maikaʻi loa, akā pono ia i ka hoʻonohonoho pono ʻana e pale i ka overcorrection.
E haʻi mau i kāu mea mālama ola e pili ana i nā lāʻau lapaʻau paʻa ʻana o ka ʻōpū āu e hoʻohana nei, me nā lāʻau lapaʻau ma luna o ka counter, nā mea hoʻohui, a me nā lāʻau lapaʻau home. Kōkua kēia iā lākou e hoʻolālā i ka hoʻolālā lapaʻau palekana a maikaʻi loa no ʻoe.
6Mpeople
Get clear medical guidance
on symptoms, medications, and lab reports.