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Chii chinonzi Naltrexone (Nzira yeIntramuscular): Zvinoshandiswa, Madosi, Migumisiro Yemuviri uye Zvimwe

Created at:1/13/2025

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Naltrexone intramuscular jekiseni imhando yejekiseni rinopiwa kamwe chete pamwedzi rinobatsira vanhu kuti varambe vakasununguka kubva mudoro kana maopioids. Mushonga uyu unoshanda nekudzivisa mibairo inofadza yezvinhu izvi muuropi hwako, zvichiita kuti zvive nyore kuchengetedza kupora kwako.

Funga nezvazvo sechidzitiro chinodzivirira chinogara kwemwedzi mumwe chete. Paunogamuchira jekiseni iri, uri kutora danho rakakosha rekupora kwenguva refu nerutsigiro rwevashandi vezvokurapa vanonzwisisa rwendo rwako.

Chii chinonzi Naltrexone Intramuscular Jekiseni?

Naltrexone intramuscular jekiseni imhando ye naltrexone inoshanda kwenguva refu inopiwa sejekiseni mumhasuru yako kamwe chete pamwedzi. Kusiyana nemapiritsi ezuva nezuva, jekiseni iri rinopa mazinga emishonga akagadzikana mumuviri wako kwemazuva anenge makumi matatu.

Mushonga uyu unopiwa nachiremba munzvimbo yekiriniki. Izvi zvinovimbisa kuti unogamuchira madosi akakodzera uye kutariswa kwezvokurapa kwakakodzera panguva yekurapa kwako.

Nzvimbo yejekiseni inowanzoita mhasuru yako yegumbo, uko mushonga unoburitswa zvishoma nezvishoma nekufamba kwenguva. Kuburitswa uku kunobatsira kuchengetedza dziviriro yakagadzikana kubva kune doro uye opioid effects.

Chii chinonzi Naltrexone chinoshandiswa?

Naltrexone intramuscular jekiseni rinonyanya kurapa dambudziko rekushandisa doro uye dambudziko rekushandisa opioid muvanhu vakuru. Yakagadzirirwa zvakananga vanhu vakasununguka kare uye vanoda kuchengetedza kupora kwavo.

Kune dambudziko rekushandisa doro, mushonga uyu unobatsira kuderedza chido uye unoita kuti kunwa kuve kushoma. Vanhu vazhinji vanozviwana zviri nyore kutevedzera zvinangwa zvavo zvekuzvidzora kana vaine rutsigiro urwu rwemwedzi.

Pakurapa dambudziko rekushandisa opioid, naltrexone inodzivisa mhedzisiro ye euphoric yeopioids senge heroin, mishonga yekurwadziwa yakanyorwa, uye fentanyl. Zvisinei, unofanira kunge wakasununguka zvachose kubva kumaopioids kwemazuva anenge 7-10 usati watanga kurapwa.

Chiremba wako angangofungawo mushonga uyu kana wakatadza kuyeuka kutora mapiritsi e naltrexone ezuva nezuva. Jekiseni remwedzi rinobvisa sarudzo yezuva nezuva yekutevedzera mushonga.

Naltrexone Inoshanda Sei?

Naltrexone inoshanda nekudzivisa maopioid receptors muuropi hwako, ayo ari ma receptors mamwechete ayo doro nemaopioid anotarisira kugadzira mhedzisiro yawo yekupa mubairo. Izvi zvinoita kuti ive mushonga wakasimba zvishoma unopa dziviriro yakavimbika.

Paunonwa doro kana kushandisa maopioid uchiita naltrexone, hauzonzwe manzwiro anowanzoita anofadza. Panzvimbo pezvo, zvinhu izvi zvinova zvisingashande pakugadzira euphoria kana kuzorora.

Mushonga haukuiti kuti unzwe kurwara kana kusanzwa zvakanaka paunosangana nezvinhu izvi. Inongobvisa ruzivo runopa mubairo runowanzoita kuti uenderere mberi nekushandisa.

Iyi mhedzisiro yekudzivisa inogara kwemwedzi wese pakati pejekiseni. Maopioid receptors muuropi hwako anoramba akabatwa ne naltrexone, achipa dziviriro inogara kunyangwe uine nguva dzekushaya simba kana kuda zvakanyanya.

Ndinofanira Kutora Sei Naltrexone Intramuscular Injection?

Uchagamuchira jekiseni rako re naltrexone muhofisi yachiremba wako kana kiriniki kamwe chete muna vhiki ina. Mupi wehutano achakupa jekiseni mumhasuru yegumbo rako, achichinjana mativi nejekiseni rega rega.

Usati waenda kumusangano wako, unogona kudya zvakajairika uye haufanire kudzivisa chero chikafu chipi zvacho. Zvisinei, kupfeka mbatya dzakasununguka kunogona kuita kuti maitiro ejekiseni ave nyore.

Jekiseni pacharo rinotora maminitsi mashoma chete, kunyangwe iwe ungada kugara kwenguva pfupi yekucherechedza. Mamwe makiriniki anoda kuongorora varwere kwemaminitsi gumi nemashanu kusvika makumi matatu mushure mejekiseni kuti ave nechokwadi chekuti hapana maitiro ekukurumidza anoitika.

Uchada kuronga musangano wako unotevera usati wabva kukiriniki. Kuchengeta chirongwa chemwedzi chinogara kunobatsira kuchengetedza mazinga emushonga akagadzikana muhurongwa hwako.

Ndingatora Naltrexone Kwenguva Yakareba Sei?

Vanhu vazhinji vanoramba vachitora majekiseni e naltrexone kwemwedzi inenge 6-12, kunyangwe vamwe vachibatsirwa nekutora kwenguva refu. Chiremba wako achashanda newe kuti aone kuti inguva yakareba sei zvichienderana nekufambira mberi kwako mukupora.

Kureba kwenguva yekurapa kunowanzoenderana nemamiriro ako, rutsigiro rwaunahwo, uye kuti uri kubata sei kupora kwako. Vamwe vanhu vanoona kuti vanoda rutsigiro rwekuenderera mberi kwemakore akati wandei, asi vamwe vanogona kuchinjira kune dzimwe nzira dzekurapa.

Mupi wako wehutano achatarisa kufambira mberi kwako nguva dzose uye achakurukura kana kuenderera mberi nekurapa kuchinzwisisika mumamiriro ako ezvinhu. Hurukuro idzi dzinowanzoitika mwedzi mitatu yega yega panguva yekugadzwa kwako kwenguva dzose.

Rangarira kuti kumisa naltrexone kunofanirwa kuve chisarudzo chakarongeka chinoitwa nekutungamirirwa nachiremba wako. Kumisa kurapwa kamwe kamwe kunogona kukusiya uchitambura nekudzokera kumashure usina masisitimu akakodzera ekutsigira.

Ndezvipi Zvakaipa ZveNaltrexone?

Vanhu vazhinji vanoshivirira majekiseni e naltrexone zvakanaka, asi unogona kusangana nezvimwe zvinokonzeresa, kunyanya mumavhiki mashoma ekutanga. Zvinhu izvi zvinowanzoitika uye zvinowanzoita nani muviri wako uchigadzirisa mushonga.

Heano mativi akajairika aunogona kuona:

  • Maitiro ekupinza senge kurwadziwa, kuzvimba, kana kutsvuka
  • Nausea kana dumbu rinogumbura
  • Musoro
  • Dizziness kana kuneta
  • Kutambudzika kurara
  • Kuderera kwechido
  • Kurwadziwa kwemhasuru kana majoini

Izvi zvinowanzoitika zvinokonzeresa zvinowanzoitika mazuva mashoma kusvika vhiki mushure mejekiseni rega rega. Vanhu vazhinji vanozviwana zvichishiviririka uye zvichibata nekuyera nyore nyore.

Zvisingawanzoitiki asi zvakanyanya kukomba zvinokonzeresa zvinogona kuitika dzimwe nguva, uye unofanirwa kubata chiremba wako kana ukaona chero zviratidzo zvinonetsa:

  • Kusagadzikana kwakanyanya panzvimbo yekujowa pamwe nekurwadziwa kana kupisa zvichikwira
  • Zviratidzo zvekuora mwoyo kana shanduko dzemanzwiro
  • Manyoka akanyanya kana kurutsa
  • Kuneta kana kushaya simba zvisingaite
  • Kurwadziwa mudumbu kana kusagadzikana

Mhedzisiro isingawanzoitiki asi yakakomba inosanganisira matambudziko echiropa, kunyangwe izvi zvisingawanzoitiki nemhando yekujowa. Chiremba wako achatarisa kushanda kwechiropa chako kuburikidza nemiedzo yeropa nguva nenguva.

Kazhinji, vamwe vanhu vanowana mhinduro dzakanyanya dzekurwara kune naltrexone. Zviratidzo zvinosanganisira kuoma kufema, kuzvimba kwechiso kana huro, kana rash yakapararira. Izvi zvinoda kutariswa kwekurapa nekukurumidza.

Ndiani Asingafaniri Kutora Naltrexone?

Naltrexone haina kuchengeteka kune vese, uye mamiriro akati wandei anoita kuti mushonga uyu usakodzere kana kuve nenjodzi. Chiremba wako achanyatsoongorora nhoroondo yako yekurapa usati wanyora mushonga uyu.

Haufaniri kuwana majekiseni e naltrexone kana iwe:

  • Parizvino uri kushandisa maopioids kana usati wava opioid-free kwemazuva angangoita 7-10
  • Une chirwere chechiropa chakanyanya kana kutadza kwechiropa
  • Une allergic ku naltrexone kana chero zvinhu zviri mujekiseni
  • Une pamuviri kana kuyamwisa
  • Une chirwere cheitsvo chakanyanya

Chiremba wako achashandisawo chenjedzo yakawedzerwa kana uine mamwe mamiriro ehutano anoda kutariswa zvakanyanya panguva yekurapa.

Vanhu vane matambudziko echiropa akapfava vangave vachiri vakwikwidzi vekurapa, asi vachada kutariswa kazhinji kuburikidza nemiedzo yeropa. Chiremba wako achayerera mabhenefiti achipesana nenjodzi mumamiriro ezvinhu aya.

Kana iwe uri kutora mishonga yeopioid yekurapa kurwadziwa, uchada kushanda nachiremba vako kuti vagadzire imwe nzira yekurapa kurwadziwa usati watanga naltrexone.

Mazita eNaltrexone Brand

Zita rinowanzozivikanwa re naltrexone intramuscular injection ndiVivitrol. Iyi ndiyo vhezheni iyo vanachiremba vazhinji vanonyora uye makambani einishuwarenzi anowanzo kufukidza.

Vivitrol ine 380 mg ye naltrexone mukati mejekiseni rega rega remwedzi. Mushonga uyu unouya semupfu uyo vanachiremba vako vanosanganisa nemvura yakakosha vasati vakupa jekiseni.

Mamwe makambani emishonga anogona kugadzira mamwe mafomu e naltrexone inotora nguva refu, asi Vivitrol inoramba iri iyo yakanyanya kudzidzwa uye yakanyorwa. Chiremba wako anogona kutanga neiyi nzira yakagadzirwa zvakanaka.

Zvimwe Zvinogona Kushandiswa Panzvimbo peNaltrexone

Mishonga yakati wandei inogona kubatsira ne dambudziko rekushandisa doro kana maopioid kana naltrexone isiri iyo yakakunakira. Chiremba wako anogona kukurukura sarudzo idzi zvichienderana nezvido zvako uye mamiriro ako.

Kune dambudziko rekushandisa doro, zvimwe zvinogona kushandiswa zvinosanganisira acamprosate, iyo inobatsira kuderedza chido, uye disulfiram, iyo inokonzera maitiro asingafadzi kana iwe uchinwa. Vamwe vanhu vanobatsirwawo ne topiramate kana gabapentin.

Kune dambudziko rekushandisa opioid, buprenorphine uye methadone ndizvo zvimwe zvinogona kushandiswa zvinobudirira. Mishonga iyi inoshanda zvakasiyana ne naltrexone nekushandisa zvishoma maopioid receptors panzvimbo yekuvharisa zvachose.

Vamwe vanhu vanoita zviri nani ne naltrexone yemumuromo yezuva nezuva kana vasingade kuwana majekiseni emwedzi. Vamwe vangabatsirwa nenzira dzakasiyana dzinosanganisira mazano, mapoka ekutsigira, uye shanduko dzemararamiro.

Naltrexone iri nani here pane Buprenorphine?

Naltrexone ne buprenorphine zvinoshanda pakurapa dambudziko rekushandisa opioid, asi zvinoshanda nenzira dzakasiyana uye zvakakodzera vanhu vakasiyana. Hapana mushonga wakanyanya "kunaka" pane mumwe.

Naltrexone inodzivisa zvachose mhedzisiro yeopioid, iyo vamwe vanhu vanosarudza nekuti haikonzeri kuvimba kwemuviri. Zvisinei, unofanira kunge usina zvachose maopioid usati watanga kurapwa, izvo zvinogona kuva zvakaoma.

Buprenorphine inoshandisa zvishoma opioid receptors, izvo zvinobatsira kudzora zviratidzo zvekusiyana uye zvishuvo ukuwo ichidzivirira mhedzisiro yeimwe opioids. Unogona kutanga mushonga uyu uchiri kusangana nekusiyana, zvichiita kuti kuchinja kuve nyore.

Chiremba wako achakubatsira kusarudza zvichienderana nemamiriro ako ega, kusanganisira kuti wakareba sei usina kunwa, rutsigiro rwako, uye zvaunofarira pachako nezve nzira dzekurapa.

Mibvunzo Inowanzo Bvunzwa Nezve Naltrexone

Q1. Naltrexone Yakachengeteka Kune Vanhu Vane Kuora Mwoyo Here?

Naltrexone inogona kushandiswa zvakachengeteka muvanhu vane kuora mwoyo, asi inoda kutariswa zvakanyanya. Vamwe vanhu vanosangana nekuchinja kwemanzwiro pavanotanga naltrexone, saka chiremba wako achada kutevera hutano hwako hwepfungwa zvakanyanya.

Kana uri kutora antidepressants, naltrexone kazhinji haipindire nemishonga iyi. Zvisinei, chiremba wako angachinja kurapwa kwako kwekuora mwoyo kuti ave nechokwadi chekuti uri kuwana hanya yakanakisisa kune zvese zvirwere.

Zvakakosha kuti uudze mupi wako wehutano nezve chero nhoroondo yekuora mwoyo kana pfungwa dzekuzviuraya. Vanogona kupa rutsigiro rwakawedzerwa uye kutariswa panguva yekurapa kwako.

Q2. Ndoitei Kana Ndikashandisa Naltrexone Yakawandisa Netsaona?

Sezvo naltrexone ichipiwa sejojo remwedzi nemapi wemishonga, overdose netsaona haisi kazhinji. Mushonga unoyereswa zvakanyanya uye unopiwa munzvimbo dzekiriniki.

Kana iwe ukawana naltrexone yakawandisa, unogona kusangana nemhedzisiro yakanyanya senausea, dzungu, kana kurwadziwa nemusoro. Bata chiremba wako nekukasira kana iwe uchitenda kuti wakagamuchira dose isiriyo.

Chinhu chakanyanya kukosha ndechitsvaga rubatsiro rwekurapa nekukasira. Mupi wako wehutano anogona kukutarisa kune chero matambudziko uye kupa rutsigiro rwekuchengetedza kana zvichidikanwa.

Q3. Ndoitei Kana Ndikakanganwa Dose yeNaltrexone?

Kana ukasavaka jekiseni rako remwedzi nemwedzi re naltrexone, taura nachiremba wako nekukurumidza sezvinobvira kuti urongezve. Zvinhu zvinodzivirira zve mushonga zvinotanga kupera mushure memazuva anenge 30.

Usamirira kusvika nguva yako inotevera yakarongwa kana wakatadza kare. Chiremba wako angada kukuona nekukurumidza kuti uchengetedze kurapwa nguva dzose uye kukurukura chero matambudziko auri kusangana nawo.

Kutadza mishonga kunogona kuwedzera njodzi yako yekudzokera kumashure, saka zvakakosha kuti udzokere munzira nekukurumidza. Chikwata chako chehutano chinogona kukubatsira kugadzira nzira dzekuyeuka misangano yeramangwana.

Q4. Ndingamira Rini Kutora Naltrexone?

Sarudzo yekumisa naltrexone inofanira kugara ichiitwa nekutungamirirwa nachiremba wako. Vanhu vazhinji vanoenderera mberi nekurapwa kwemwedzi inenge 6-12, kunyangwe vamwe vachibatsirwa nenguva refu.

Chiremba wako achafunga nezvezvinhu zvakaita sekufambira mberi kwako mukupora, tsigiro, uye zvinangwa zvako pachako paunenge uchikurukura kumisa. Vanogona kukurudzira kuparadzira zvishoma nezvishoma majekiseni kana kuchinjira kune dzimwe nzira dzekutsigira.

Usati wamisa naltrexone, ita shuwa kuti une nzira dzakasimba dzekugadzirisa uye masisitimu ekutsigira. Chikwata chako chehutano chinogona kukubatsira kugadzira chirongwa chakazara chekuchengetedza kupora kwako.

Q5. Ndinganwa Doro Ndiri Kutora Naltrexone?

Nepo naltrexone ichivharira mhedzisiro inobatsira ye doro, kunwa uchiri pamushonga uyu hakukurudzirwi. Mushonga unoderedza mhedzisiro inofadza ye doro, asi unogona kuramba uchisangana nekukanganiswa uye njodzi dzehutano.

Vamwe vanhu vanowana kuti doro rinonaka zvakasiyana kana risiri pa naltrexone. Izvi ndizvo chaizvo zvinoita kuti mushonga ubatsire kuderedza maitiro ekunwa nekufamba kwenguva.

Kana ukaita kunwa uchiri pa naltrexone, hauzowana buzz yenguva dzose, asi unogona kuramba uchisangana nemahangovers, kutonga kwakashata, uye mamwe matambudziko ane chekuita nedoro. Chinangwa ndechekuchengetedza kuzvidzora kwakakwana kuti uwane mhedzisiro yakanaka.

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